3NW6.A | IGF1R

General Structure Information 3nw6 IGF1R crystal structure of insulin-like growth factor 1 receptor (igf-1r-wt) complex with a carbon-linked proline isostere inhibitor (11a) 2.2Å AUTH A.J.SAMPOGNARO,M.D.WITTMAN,J.M.CARBONI,C.CHANG,A.F.GREER,AUTH 2 W.W.HURLBURT,J.S.SACK,D.M.VYASTITL PROLINE ISOSTERES IN A SERIES OF 2,4-DISUBSTITUTEDTITL 2 PYRROLO[1,2-F][1,2,4]TRIAZINE INHIBITORS OF IGF-1R KINASETITL 3 AND IR KINASE.REF BIOORG.MED.CHEM.LETT. V. 20 5027 2010REFN ISSN 0960-894XPMID 20675137DOI 10.1016/J.BMCL.2010.07.045 Variant Set […]

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