4IAR.A | HTR1B

General Structure Information 4iar HTR1B crystal structure of the chimeric protein of 5-ht1b-bril in complex with ergotamine (psi community target) 2.7Å AUTH C.WANG,Y.JIANG,J.MA,H.WU,D.WACKER,V.KATRITCH,G.W.HAN,W.LIU,AUTH 2 X.P.HUANG,E.VARDY,J.D.MCCORVY,X.GAO,X.E.ZHOU,K.MELCHER,AUTH 3 C.ZHANG,F.BAI,H.YANG,L.YANG,H.JIANG,B.L.ROTH,V.CHEREZOV,AUTH 4 R.C.STEVENS,H.E.XUTITL STRUCTURAL BASIS FOR MOLECULAR RECOGNITION AT SEROTONINTITL 2 RECEPTORS.REF SCIENCE V. 340 610 2013REFN ISSN 0036-8075PMID 23519210DOI 10.1126/SCIENCE.1232807 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

See Details
2KOE.A | CNR1

General Structure Information 2koe CNR1 human cannabinoid receptor 1 – helix 7/8 peptide -1.0Å AUTH S.TYUKHTENKO,E.K.TIBURU,L.DESHMUKH,O.VINOGRADOVA,AUTH 2 D.R.JANERO,A.MAKRIYANNISTITL NMR SOLUTION STRUCTURE OF HUMAN CANNABINOIDTITL 2 RECEPTOR-1 HELIX 7/8 PEPTIDE: CANDIDATETITL 3 ELECTROSTATIC INTERACTIONS AND MICRODOMAINTITL 4 FORMATION.REF BIOCHEM.BIOPHYS.RES.COMMUN. V. 390 441 2009REFN ISSN 0006-291XPMID 19766594DOI 10.1016/J.BBRC.2009.09.053 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

See Details
3QAK.A | ADORA2A

General Structure Information 3qak ADORA2A agonist bound structure of the human adenosine a2a receptor 2.71Å AUTH F.XU,H.WU,V.KATRITCH,G.W.HAN,K.A.JACOBSON,Z.G.GAO,AUTH 2 V.CHEREZOV,R.C.STEVENSTITL STRUCTURE OF AN AGONIST-BOUND HUMAN A2A ADENOSINE RECEPTOR.REF SCIENCE V. 332 322 2011REFN ISSN 0036-8075PMID 21393508DOI 10.1126/SCIENCE.1202793 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

See Details
3G04.C | TSHR

General Structure Information 3g04 TSHR crystal structure of the tsh receptor in complex with a thyroid- stimulating autoantibody 2.55Å AUTH J.SANDERS,D.Y.CHIRGADZE,P.SANDERS,S.BAKER,A.SULLIVAN,AUTH 2 A.BHARDWAJA,J.BOLTON,M.REEVE,N.NAKATAKE,M.EVANS,T.RICHARDS,AUTH 3 M.POWELL,R.N.MIGUEL,T.L.BLUNDELL,J.FURMANIAK,B.R.SMITHTITL CRYSTAL STRUCTURE OF THE TSH RECEPTOR IN COMPLEX WITH ATITL 2 THYROID-STIMULATING AUTOANTIBODYREF THYROID V. 17 395 2007REFN ISSN 1050-7256PMID 17542669DOI 10.1089/THY.2007.0034 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

See Details
2L64.A | GCG

General Structure Information 2l64 GCG nmr solution structure of glp-2 in dhpc micelles -1.0Å AUTH K.C.VENNETI,C.M.HEWAGETITL CONFORMATIONAL AND MOLECULAR INTERACTION STUDIES OFTITL 2 GLUCAGON-LIKE PEPTIDE-2 WITH ITS N-TERMINAL EXTRACELLULARTITL 3 RECEPTOR DOMAIN.REF FEBS LETT. V. 585 346 2011REFN ISSN 0014-5793PMID 21167157DOI 10.1016/J.FEBSLET.2010.12.011 Variant Set Distributions Mapped Variants

See Details
3N7P.D | RAMP1

General Structure Information 3n7p RAMP1 crystal structure of the ectodomain complex of the cgrp receptor, a class-b gpcr, reveals the site of drug antagonism 2.8Å AUTH E.TER HAAR,C.M.KOTH,N.ABDUL-MANAN,L.SWENSON,J.T.COLL,AUTH 2 J.A.LIPPKE,C.A.LEPRE,M.GARCIA-GUZMAN,J.M.MOORETITL CRYSTAL STRUCTURE OF THE ECTODOMAIN COMPLEX OF THE CGRPTITL 2 RECEPTOR, A CLASS-B GPCR, REVEALS THE SITE OF DRUGTITL 3 ANTAGONISM.REF STRUCTURE V. 18 1083 […]

See Details