3E37.A | FNTA

General Structure Information 3e37 FNTA protein farnesyltransferase complexed with bisubstrate ethylenediamine scaffold inhibitor 5 1.8Å AUTH M.A.HAST,S.FLETCHER,C.G.CUMMINGS,E.E.PUSATERI,AUTH 2 M.A.BLASKOVICH,K.RIVAS,M.H.GELB,W.C.VAN VOORHIS,AUTH 3 S.M.SEBTI,A.D.HAMILTON,L.S.BEESETITL STRUCTURAL BASIS FOR BINDING AND SELECTIVITY OFTITL 2 ANTIMALARIAL AND ANTICANCER ETHYLENEDIAMINETITL 3 INHIBITORS TO PROTEIN FARNESYLTRANSFERASE.REF CHEM.BIOL. V. 16 181 2009REFN ISSN 1074-5521PMID 19246009DOI 10.1016/J.CHEMBIOL.2009.01.014 Variant Set Distributions Ripley’s K Analysis Plots […]

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3WEF.C | FDFT1

General Structure Information 3wef FDFT1 crystal structure of the human squalene synthase in complex with farnesyl thiopyrophosphate 2.35Å AUTH C.I.LIU,W.Y.JENG,W.J.CHANG,M.F.SHIH,T.P.KO,A.H.J.WANGTITL STRUCTURAL INSIGHTS INTO THE CATALYTIC MECHANISM OF HUMANTITL 2 SQUALENE SYNTHASEREF ACTA CRYSTALLOGR.,SECT.D V. 70 231 2014REFN ISSN 0907-4449DOI 10.1107/S1399004713026230 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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