2YGQ.A | WIF1

General Structure Information 2ygq WIF1 wif domain-epidermal growth factor (egf)-like domains 1-3 of human wnt inhibitory factor 1 in complex with 1,2-dipalmitoylphosphatidylcholine 3.95Å AUTH T.MALINAUSKAS,A.R.ARICESCU,W.LU,C.SIEBOLD,E.Y.JONESTITL MODULAR MECHANISM OF WNT SIGNALING INHIBITION BY WNTTITL 2 INHIBITORY FACTOR 1REF NAT.STRUCT.MOL.BIOL. V. 18 886 2011REFN ISSN 1545-9993PMID 21743455DOI 10.1038/NSMB.2081 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1L2J.B | ESR2

General Structure Information 1l2j ESR2 human estrogen receptor beta ligand-binding domain in complex with (r, r)-5,11-cis-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol 2.95Å AUTH A.K.SHIAU,D.BARSTAD,J.T.RADEK,M.J.MEYERS,K.W.NETTLES,AUTH 2 B.S.KATZENELLENBOGEN,J.A.KATZENELLENBOGEN,D.A.AGARD,AUTH 3 G.L.GREENETITL STRUCTURAL CHARACTERIZATION OF A SUBTYPE-SELECTIVE LIGANDTITL 2 REVEALS A NOVEL MODE OF ESTROGEN RECEPTOR ANTAGONISM.REF NAT.STRUCT.BIOL. V. 9 359 2002REFN ISSN 1072-8368PMID 11953755 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1VJB.B | ESRRG

General Structure Information 1vjb ESRRG crystal structure of the ligand-binding domain of the estrogen-related receptor gamma in complex with 4- hydroxytamoxifen 3.2Å AUTH H.GRESCHIK,R.FLAIG,J.P.RENAUD,D.MORASTITL STRUCTURAL BASIS FOR THE DEACTIVATION OF THETITL 2 ESTROGEN-RELATED RECEPTOR {GAMMA} BYTITL 3 DIETHYLSTILBESTROL OR 4-HYDROXYTAMOXIFEN ANDTITL 4 DETERMINANTS OF SELECTIVITY.REF J.BIOL.CHEM. V. 279 33639 2004REFN ISSN 0021-9258PMID 15161930DOI 10.1074/JBC.M402195200 Variant […]

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3N7P.D | RAMP1

General Structure Information 3n7p RAMP1 crystal structure of the ectodomain complex of the cgrp receptor, a class-b gpcr, reveals the site of drug antagonism 2.8Å AUTH E.TER HAAR,C.M.KOTH,N.ABDUL-MANAN,L.SWENSON,J.T.COLL,AUTH 2 J.A.LIPPKE,C.A.LEPRE,M.GARCIA-GUZMAN,J.M.MOORETITL CRYSTAL STRUCTURE OF THE ECTODOMAIN COMPLEX OF THE CGRPTITL 2 RECEPTOR, A CLASS-B GPCR, REVEALS THE SITE OF DRUGTITL 3 ANTAGONISM.REF STRUCTURE V. 18 1083 […]

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