2J0F.A | TYMP

General Structure Information 2j0f TYMP structural basis for non-competitive product inhibition in human thymidine phosphorylase: implication for drug design 2.31Å AUTH K.EL OMARI,A.BRONCKAERS,S.LIEKENS,M.PEREZ-PEREZ,AUTH 2 J.BALZARINI,D.K.STAMMERSTITL STRUCTURAL BASIS FOR NON-COMPETITIVE PRODUCTTITL 2 INHIBITION IN HUMAN THYMIDINE PHOSPHORYLASE:TITL 3 IMPLICATIONS FOR DRUG DESIGN.REF BIOCHEM.J. V. 399 199 2006REFN ISSN 0264-6021PMID 16803458DOI 10.1042/BJ20060513 Variant Set Distributions Ripley’s K […]

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3HNG.A | FLT1

General Structure Information 3hng FLT1 crystal structure of vegfr1 in complex with n-(4-chlorophenyl)-2- ((pyridin-4-ylmethyl)amino)benzamide 2.7Å AUTH L.TRESAUGUES,A.ROOS,C.H.ARROWSMITH,H.BERGLUND,C.BOUNTRA,AUTH 2 R.COLLINS,A.M.EDWARDS,S.FLODIN,A.FLORES,S.GRASLUND,AUTH 3 M.HAMMARSTROM,A.JOHANSSON,I.JOHANSSON,T.KARLBERG,AUTH 4 T.KOTENYOVA,M.MOCHE,T.NYMAN,C.PERSSON,T.KRAGH-NIELSEN,AUTH 5 A.KOTZCH,J.SAGEMARK,H.SCHUELER,P.SCHUTZ,M.I.SIPONEN,AUTH 6 L.SVENSSON,A.G.THORSELL,S.VAN DER BERG,J.WEIGELT,M.WELIN,AUTH 7 M.WISNIEWSKA,P.NORDLUNDTITL CRYSTAL STRUCTURE OF VEGFR1 IN COMPLEX WITHTITL 2 N-(4-CHLOROPHENYL)-2-((PYRIDIN-4-YLMETHYL)AMINO)BENZAMIDEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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3FJI.A | FGF1

General Structure Information 3fji FGF1 crystal structure of k12v/c83i/c117v mutant of human acidic fibroblast growth factor 2.55Å AUTH J.LEE,M.BLABERTITL STRUCTURAL BASIS OF CONSERVED CYSTEINE IN THETITL 2 FIBROBLAST GROWTH FACTOR FAMILY: EVIDENCE FOR ATITL 3 VESTIGIAL HALF-CYSTINE.REF J.MOL.BIOL. V. 393 128 2009REFN ISSN 0022-2836PMID 19683004DOI 10.1016/J.JMB.2009.08.007 Variant Set Distributions Mapped Variants

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2XV7.A | FIGF

General Structure Information 2xv7 FIGF crystal structure of vascular endothelial growth factor d 2.9Å AUTH V.M.LEPPANEN,M.JELTSCH,A.ANISIMOV,D.TVOROGOV,K.AHO,AUTH 2 N.KALKKINEN,P.TOIVANEN,S.YLA-HERTTUALA,K.BALLMER-HOFER,AUTH 3 K.ALITALOTITL STRUCTURAL DETERMINANTS OF VASCULAR ENDOTHELIAL GROWTHTITL 2 FACTOR-D – RECEPTOR BINDING AND SPECIFICITY.REF BLOOD V. 117 1507 2011REFN ISSN 0006-4971PMID 21148085DOI 10.1182/BLOOD-2010-08-301549 Variant Set Distributions Mapped Variants

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2QQM.A | NRP1

General Structure Information 2qqm NRP1 crystal structure of the a2b1b2 domains from human neuropilin-1 2.0Å AUTH B.A.APPLETON,P.WU,J.MALONEY,J.YIN,W.C.LIANG,S.STAWICKI,AUTH 2 K.MORTARA,K.K.BOWMAN,J.M.ELLIOTT,W.DESMARAIS,J.F.BAZAN,AUTH 3 A.BAGRI,M.TESSIER-LAVIGNE,A.W.KOCH,Y.WU,R.J.WATTS,C.WIESMANNTITL STRUCTURAL STUDIES OF NEUROPILIN/ANTIBODY COMPLEXES PROVIDETITL 2 INSIGHTS INTO SEMAPHORIN AND VEGF BINDINGREF EMBO J. V. 26 4902 2007REFN ISSN 0261-4189PMID 17989695DOI 10.1038/SJ.EMBOJ.7601906 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic […]

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1Z3S.B | ANGPT2

General Structure Information 1z3s ANGPT2 angiopoietin-2 receptor binding domain 2.35Å AUTH W.A.BARTON,D.TZVETKOVA,D.B.NIKOLOVTITL STRUCTURE OF THE ANGIOPOIETIN-2 RECEPTOR BINDINGTITL 2 DOMAIN AND IDENTIFICATION OF SURFACES INVOLVED INTITL 3 TIE2 RECOGNITION.REF STRUCTURE V. 13 825 2005REFN ISSN 0969-2126PMID 15893672DOI 10.1016/J.STR.2005.03.009 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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