1KSN.B | F10

General Structure Information 1ksn F10 crystal structure of human coagulation factor xa complexed with fxv673 2.1Å AUTH K.R.GUERTIN,C.J.GARDNER,S.I.KLEIN,A.L.ZULLI,AUTH 2 M.CZEKAJ,Y.GONG,A.P.SPADA,D.L.CHENEY,S.MAIGNAN,AUTH 3 J.P.GUILLOTEAU,K.D.BROWN,D.J.COLUSSI,V.CHU,AUTH 4 C.L.HERAN,S.R.MORGAN,R.G.BENTLEY,C.T.DUNWIDDIE,AUTH 5 R.J.LEADLEY,H.W.PAULSTITL OPTIMIZATION OF THE BETA-AMINOESTER CLASS OFTITL 2 FACTOR XA INHIBITORS. PART 2: IDENTIFICATION OFTITL 3 FXV673 AS A POTENT AND SELECTIVE INHIBITOR WITHTITL 4 EXCELLENT IN VIVO ANTICOAGULANT ACTIVITY.REF […]

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1QUB.A | APOH

General Structure Information 1qub APOH crystal structure of the glycosylated five-domain human beta2- glycoprotein i purified from blood plasma 2.7Å AUTH B.BOUMA,P.G.DE GROOT,J.M.VAN DEN ELSEN,R.B.RAVELLI,AUTH 2 A.SCHOUTEN,M.J.SIMMELINK,R.H.DERKSEN,J.KROON,P.GROSTITL ADHESION MECHANISM OF HUMAN BETA(2)-GLYCOPROTEIN I TOTITL 2 PHOSPHOLIPIDS BASED ON ITS CRYSTAL STRUCTURE.REF EMBO J. V. 18 5166 1999REFN ISSN 0261-4189PMID 10508150DOI 10.1093/EMBOJ/18.19.5166 Variant Set Distributions Ripley’s […]

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1NFA.A | NFATC1

General Structure Information 1nfa NFATC1 human transcription factor nfatc dna binding domain, nmr, 10 structures -1.0Å AUTH S.A.WOLFE,P.ZHOU,V.DOTSCH,L.CHEN,A.YOU,S.N.HO,AUTH 2 G.R.CRABTREE,G.WAGNER,G.L.VERDINETITL UNUSUAL REL-LIKE ARCHITECTURE IN THE DNA-BINDINGTITL 2 DOMAIN OF THE TRANSCRIPTION FACTOR NFATC.REF NATURE V. 385 172 1997REFN ISSN 0028-0836PMID 8990122DOI 10.1038/385172A0 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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1UMK.A | CYB5R3

General Structure Information 1umk CYB5R3 the structure of human erythrocyte nadh-cytochrome b5 reductase 1.75Å AUTH S.BANDO,T.TAKANO,T.YUBISUI,K.SHIRABE,M.TAKESHITA,AUTH 2 A.NAKAGAWATITL STRUCTURE OF HUMAN ERYTHROCYTE NADH-CYTOCHROME B5TITL 2 REDUCTASE.REF ACTA CRYSTALLOGR.,SECT.D V. 60 1929 2004REFN ISSN 0907-4449PMID 15502298DOI 10.1107/S0907444904020645 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1BIK.A | AMBP

General Structure Information 1bik AMBP x-ray structure of bikunin from the human inter-alpha-inhibitor complex 2.5Å AUTH Y.XU,P.D.CARR,J.M.GUSS,D.L.OLLISTITL THE CRYSTAL STRUCTURE OF BIKUNIN FROM THETITL 2 INTER-ALPHA-INHIBITOR COMPLEX: A SERINE PROTEASE INHIBITORTITL 3 WITH TWO KUNITZ DOMAINS.REF J.MOL.BIOL. V. 276 955 1998REFN ISSN 0022-2836PMID 9566199DOI 10.1006/JMBI.1997.1582 Variant Set Distributions Mapped Variants

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1J8K.A | FN1

General Structure Information 1j8k FN1 nmr structure of the fibronectin eda domain, nmr, 20 structures -1.0Å AUTH T.NIIMI,M.OSAWA,N.YAMAJI,K.YASUNAGA,H.SAKASHITA,AUTH 2 T.MASE,A.TANAKA,S.FUJITATITL NMR STRUCTURE OF HUMAN FIBRONECTIN EDA.REF J.BIOMOL.NMR V. 21 281 2001REFN ISSN 0925-2738PMID 11775745DOI 10.1023/A:1012947209393 Variant Set Distributions Mapped Variants

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4NQK.C | DDX58

General Structure Information 4nqk DDX58 structure of an ubiquitin complex 3.7Å AUTH A.PEISLEY,B.WU,H.XU,Z.J.CHEN,S.HURTITL STRUCTURAL BASIS FOR UBIQUITIN-MEDIATED ANTIVIRAL SIGNALTITL 2 ACTIVATION BY RIG-I.REF NATURE V. 509 110 2014REFN ISSN 0028-0836PMID 24590070DOI 10.1038/NATURE13140 Variant Set Distributions Mapped Variants

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3F6U.H | PROC

General Structure Information 3f6u PROC crystal structure of human activated protein c (apc) complexed with ppack 2.8Å AUTH A.E.SCHMIDT,K.PADMANABHAN,M.C.UNDERWOOD,W.BODE,T.MATHER,AUTH 2 S.P.BAJAJTITL THERMODYNAMIC LINKAGE BETWEEN THE S1 SITE, THE NA+ SITE, ANDTITL 2 THE CA2+ SITE IN THE PROTEASE DOMAIN OF HUMAN ACTIVATEDTITL 3 PROTEIN C (APC).REF J.BIOL.CHEM. V. 277 28987 2002REFN ISSN 0021-9258PMID 12029084DOI 10.1074/JBC.M201892200 […]

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1AS4.A | SERPINA3

General Structure Information 1as4 SERPINA3 cleaved antichymotrypsin a349r 2.1Å AUTH C.M.LUKACS,H.RUBIN,D.W.CHRISTIANSONTITL ENGINEERING AN ANION-BINDING CAVITY INTITL 2 ANTICHYMOTRYPSIN MODULATES THE SPRING-LOADEDTITL 3 SERPIN-PROTEASE INTERACTION.REF BIOCHEMISTRY V. 37 3297 1998REFN ISSN 0006-2960PMID 9521649DOI 10.1021/BI972359E Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3LC4.A | CYP2E1

General Structure Information 3lc4 CYP2E1 human cytochrome p450 2e1 in complex with omega-imidazolyl-dodecanoic acid 3.1Å AUTH P.R.PORUBSKY,K.P.BATTAILE,E.E.SCOTTTITL HUMAN CYTOCHROME P450 2E1 STRUCTURES WITH FATTY ACID ANALOGSTITL 2 REVEAL A PREVIOUSLY UNOBSERVED BINDING MODE.REF J.BIOL.CHEM. V. 285 22282 2010REFN ISSN 0021-9258PMID 20463018DOI 10.1074/JBC.M110.109017 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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