General Structure Information
| PDB ID | 4ir4 |
| HGNC Gene Label(s) | BAZ2B |
| Structure Name | crystal structure of the bromodomain of human baz2b in complex with 1- [7-(morpholin-4-yl)-1-(pyridin-2-yl)indolizin-3-yl]ethanone (gsk2834113a) |
| Resolution | 2.05Å |
| Reference | AUTH P.CHEN,A.CHAIKUAD,P.BAMBOROUGH,M.BANTSCHEFF,C.BOUNTRA,AUTH 2 C.W.CHUNG,O.FEDOROV,P.GRANDI,D.JUNG,R.LESNIAK,M.LINDON,AUTH 3 S.MULLER,M.PHILPOTT,R.PRINJHA,C.ROGERS,C.SELENSKI,C.TALLANT,AUTH 4 T.WERNER,T.M.WILLSON,S.KNAPP,D.H.DREWRYTITL DISCOVERY AND CHARACTERIZATION OF GSK2801, A SELECTIVETITL 2 CHEMICAL PROBE FOR THE BROMODOMAINS BAZ2A AND BAZ2B.REF J.MED.CHEM. 2015REFN ISSN 0022-2623PMID 25799074DOI 10.1021/ACS.JMEDCHEM.5B00209 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 114 |
| Number Of SNVs | 24 |
| Number Of Permutations | 13271 |
| Optimal Distance Threshold | 11.0 |
| K Statistic | 0.101 |
| p-value | 0.046 |