3Q2G.B | ADAMTS1

General Structure Information

PDB ID 3q2g
HGNC Gene Label(s) ADAMTS1
Structure Name adamts1 in complex with a novel n-hydroxyformamide inhibitors
Resolution 2.3Å
Reference AUTH C.DE SAVI,A.PAPE,J.G.CUMMING,A.TING,P.D.SMITH,J.N.BURROWS,AUTH 2 M.MILLS,C.DAVIES,S.LAMONT,D.MILNE,C.COOK,P.MOORE,Y.SAWYER,AUTH 3 S.GERHARDTTITL THE DESIGN AND SYNTHESIS OF NOVEL N-HYDROXYFORMAMIDETITL 2 INHIBITORS OF ADAM-TS4 FOR THE TREATMENT OF OSTEOARTHRITISREF BIOORG.MED.CHEM.LETT. V. 21 1376 2011REFN ISSN 0960-894XPMID 21300546DOI 10.1016/J.BMCL.2011.01.036

Variant Set Distributions

ExAC Variants

Number Of Residues 278
Number Of SNVs 73
Number Of Permutations 10150
Optimal Distance Threshold 12.0
K Statistic 0.096
p-value 0.511

Mapped Variants

[+] ExAC Missense Variants