General Structure Information
| PDB ID | 4mp7 |
| HGNC Gene Label(s) | PDK2 |
| Structure Name | crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor pa7 |
| Resolution | 1.8Å |
| Reference | AUTH S.C.TSO,X.QI,W.J.GUI,C.Y.WU,J.L.CHUANG,AUTH 2 I.WERNSTEDT-ASTERHOLM,L.K.MORLOCK,K.R.OWENS,P.E.SCHERER,AUTH 3 N.S.WILLIAMS,U.K.TAMBAR,R.M.WYNN,D.T.CHUANGTITL STRUCTURE-GUIDED DEVELOPMENT OF SPECIFIC PYRUVATETITL 2 DEHYDROGENASE KINASE INHIBITORS TARGETING THE ATP-BINDINGTITL 3 POCKET.REF J.BIOL.CHEM. V. 289 4432 2014REFN ISSN 0021-9258PMID 24356970DOI 10.1074/JBC.M113.533885 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 363 |
| Number Of SNVs | 75 |
| Number Of Permutations | 39435 |
| Optimal Distance Threshold | 15.0 |
| K Statistic | 0.116 |
| p-value | 0.158 |