General Structure Information
| PDB ID | 3vi8 |
| HGNC Gene Label(s) | PPARA |
| Structure Name | human pprr alpha ligand binding domain in complex with a synthetic agonist aphm13 |
| Resolution | 1.75Å |
| Reference | AUTH N.KUWABARA,T.OYAMA,D.TOMIOKA,M.OHASHI,J.YANAGISAWA,AUTH 2 T.SHIMIZU,H.MIYACHITITL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS (PPARS) HAVETITL 2 MULTIPLE BINDING POINTS THAT ACCOMMODATE LIGANDS IN VARIOUSTITL 3 CONFORMATIONS: PHENYLPROPANOIC ACID-TYPE PPAR LIGANDS BINDTITL 4 TO PPAR IN DIFFERENT CONFORMATIONS, DEPENDING ON THE SUBTYPEREF J.MED.CHEM. V. 55 893 2012REFN ISSN 0022-2623PMID 22185225DOI 10.1021/JM2014293 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 258 |
| Number Of SNVs | 52 |
| Number Of Permutations | 21595 |
| Optimal Distance Threshold | 8.0 |
| K Statistic | 0.031 |
| p-value | 0.241 |