General Structure Information
| PDB ID | 3wiy |
| HGNC Gene Label(s) | MCL1 |
| Structure Name | crystal structure of mcl-1 in complex with compound 10 |
| Resolution | 2.15Å |
| Reference | AUTH Y.TANAKA,K.AIKAWA,G.NISHIDA,M.HOMMA,S.SOGABE,S.IGAKI,AUTH 2 Y.HAYANO,T.SAMESHIMA,I.MIYAHISA,T.KAWAMOTO,M.TAWADA,Y.IMAI,AUTH 3 M.INAZUKA,N.CHO,Y.IMAEDA,T.ISHIKAWATITL DISCOVERY OF POTENT MCL-1/BCL-XL DUAL INHIBITORS BY USING ATITL 2 HYBRIDIZATION STRATEGY BASED ON STRUCTURAL ANALYSIS OFTITL 3 TARGET PROTEINS.REF J.MED.CHEM. V. 56 9635 2013REFN ISSN 0022-2623PMID 24215352DOI 10.1021/JM401170C |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 150 |
| Number Of SNVs | 38 |
| Number Of Permutations | 10028 |
| Optimal Distance Threshold | 9.0 |
| K Statistic | 0.107 |
| p-value | 0.176 |