2X2R.A | KIF11

General Structure Information

PDB ID 2x2r
HGNC Gene Label(s) KIF11
Structure Name crystal structure of human kinesin eg5 in complex with (r)-2-amino-3-((4-chlorophenyl)diphenylmethylthio)propanoic acid
Resolution 2.2Å
Reference AUTH H.Y.K.KAAN,J.WEISS,D.MENGER,V.ULAGANATHAN,K.TKOCZ,C.LAGGNER,AUTH 2 F.POPOWYCZ,B.JOSEPH,F.KOZIELSKITITL STRUCTURE-ACTIVITY RELATIONSHIP AND MULTIDRUG RESISTANCETITL 2 STUDY OF NEW S-TRITYL-L-CYSTEINE DERIVATIVES AS INHIBITORSTITL 3 OF EG5.REF J.MED.CHEM. V. 54 1576 2011REFN ISSN 0022-2623PMID 21344920DOI 10.1021/JM100991M

Variant Set Distributions

ExAC Variants

Number Of Residues 331
Number Of SNVs 37
Number Of Permutations 27166
Optimal Distance Threshold 19.0
K Statistic 0.305
p-value 0.415

Mapped Variants

[+] ExAC Missense Variants