General Structure Information
| PDB ID | 4nh9 |
| HGNC Gene Label(s) | HSP90B1 |
| Structure Name | correlation between chemotype-dependent binding conformations of hsp90 alpha/beta and isoform selectivity |
| Resolution | 2.77Å |
| Reference | AUTH J.T.ERNST,M.LIU,H.ZUCCOLA,T.NEUBERT,K.BEAUMONT,A.TURNBULL,AUTH 2 A.KALLEL,B.VOUGHT,D.STAMOSTITL CORRELATION BETWEEN CHEMOTYPE-DEPENDENT BINDINGTITL 2 CONFORMATIONS OF HSP90 ALPHA / BETA AND ISOFORMTITL 3 SELECTIVITY-IMPLICATIONS FOR THE STRUCTURE-BASED DESIGN OFTITL 4 HSP90 ALPHA / BETA SELECTIVE INHIBITORS FOR TREATINGTITL 5 NEURODEGENERATIVE DISEASES.REF BIOORG.MED.CHEM.LETT. V. 24 204 2014REFN ISSN 0960-894XPMID 24332488DOI 10.1016/J.BMCL.2013.11.036 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 214 |
| Number Of SNVs | 37 |
| Number Of Permutations | 20081 |
| Optimal Distance Threshold | 7.0 |
| K Statistic | 0.042 |
| p-value | 0.623 |