4LUO.A | RPA1

General Structure Information

PDB ID 4luo
HGNC Gene Label(s) RPA1
Structure Name fragment-based discovery of a potent inhibitor of replication protein a protein-protein interactions
Resolution 1.54Å
Reference AUTH A.O.FRANK,M.D.FELDKAMP,J.P.KENNEDY,A.G.WATERSON,N.F.PELZ,AUTH 2 J.D.PATRONE,B.VANGAMUDI,D.V.CAMPER,O.W.ROSSANESE,W.J.CHAZIN,AUTH 3 S.W.FESIKTITL DISCOVERY OF A POTENT INHIBITOR OF REPLICATION PROTEIN ATITL 2 PROTEIN-PROTEIN INTERACTIONS USING A FRAGMENT-LINKINGTITL 3 APPROACH.REF J.MED.CHEM. V. 56 9242 2013REFN ISSN 0022-2623PMID 24147804DOI 10.1021/JM401333U

Variant Set Distributions

ExAC Variants

Number Of Residues 120
Number Of SNVs 35
Number Of Permutations 8895
Optimal Distance Threshold 8.0
K Statistic 0.089
p-value 0.876

Mapped Variants

[+] ExAC Missense Variants