General Structure Information
| PDB ID | 4l3p |
| HGNC Gene Label(s) | TAB1 |
| Structure Name | crystal structure of 2-(1-benzothiophen-7-yl)-4-[1-(piperidin-4-yl)- 1h-pyrazol-4-yl]furo[2,3-c]pyridin-7-amine bound to tak1-tab1 |
| Resolution | 2.68Å |
| Reference | AUTH K.R.HORNBERGER,D.M.BERGER,A.P.CREW,H.DONG,A.KLEINBERG,AUTH 2 A.H.LI,M.R.MEDEIROS,M.J.MULVIHILL,K.SIU,J.TARRANT,J.WANG,AUTH 3 F.WENG,V.L.WILDE,M.ALBERTELLA,M.BITTNER,A.COOKE,M.J.GRAY,AUTH 4 P.MARESCA,E.MAY,P.MEYN,W.PEICK,D.ROMASHKO,M.TANOWITZ,B.TOKARTITL DISCOVERY AND OPTIMIZATION OF 7-AMINOFURO[2,3-C]PYRIDINETITL 2 INHIBITORS OF TAK1.REF BIOORG.MED.CHEM.LETT. V. 23 4517 2013REFN ISSN 0960-894XPMID 23850198DOI 10.1016/J.BMCL.2013.06.053 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 30 |
| Number Of SNVs | 11 |
| Number Of Permutations | 723 |
| Optimal Distance Threshold | 11.0 |
| K Statistic | 0.273 |
| p-value | 0.865 |