General Structure Information
| PDB ID | 4krs |
| HGNC Gene Label(s) | TNKS |
| Structure Name | tankyrase-1 complexed with small molecule inhibitor |
| Resolution | 2.29Å |
| Reference | AUTH M.D.SHULTZ,D.MAJUMDAR,D.N.CHIN,P.D.FORTIN,Y.FENG,T.GOULD,AUTH 2 C.A.KIRBY,T.STAMS,N.J.WATERS,W.SHAOTITL STRUCTURE-EFFICIENCY RELATIONSHIP OFTITL 2 [1,2,4]TRIAZOL-3-YLAMINES AS NOVEL NICOTINAMIDE ISOSTERESTITL 3 THAT INHIBIT TANKYRASES.REF J.MED.CHEM. V. 56 7049 2013REFN ISSN 0022-2623PMID 23879431DOI 10.1021/JM400826J |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 204 |
| Number Of SNVs | 41 |
| Number Of Permutations | 15253 |
| Optimal Distance Threshold | 13.0 |
| K Statistic | 0.129 |
| p-value | 0.143 |