General Structure Information
| PDB ID | 3nmq |
| HGNC Gene Label(s) | HSP90AB1 |
| Structure Name | hsp90b n-terminal domain in complex with ec44, a pyrrolo-pyrimidine methoxypyridine inhibitor |
| Resolution | 2.2Å |
| Reference | AUTH T.J.YUN,E.K.HARNING,K.GIZA,D.RABAH,P.LI,J.W.ARNDT,AUTH 2 D.LUCHETTI,M.A.BIAMONTE,J.SHI,K.LUNDGREN,A.MANNING,M.R.KEHRYTITL EC144, A SYNTHETIC INHIBITOR OF HEAT SHOCK PROTEIN 90,TITL 2 BLOCKS INNATE AND ADAPTIVE IMMUNE RESPONSES IN MODELS OFTITL 3 INFLAMMATION AND AUTOIMMUNITY.REF J.IMMUNOL. V. 186 563 2011REFN ISSN 0022-1767PMID 21131419DOI 10.4049/JIMMUNOL.1000222 |
Variant Set Distributions
ExAC Variants
| Number Of Residues | 214 |
| Number Of SNVs | 39 |
| Number Of Permutations | 12027 |
| Optimal Distance Threshold | 10.0 |
| K Statistic | 0.092 |
| p-value | 0.543 |