2A8H.A | ADAM17

General Structure Information

PDB ID 2a8h
HGNC Gene Label(s) ADAM17
Structure Name crystal structure of catalytic domain of tace with thiomorpholine sulfonamide hydroxamate inhibitor
Resolution 2.3Å
Reference AUTH J.I.LEVIN,J.M.CHEN,L.M.LAAKSO,M.DU,J.SCHMID,W.XU,AUTH 2 T.CUMMONS,J.XU,G.JIN,D.BARONE,J.S.SKOTNICKITITL ACETYLENIC TACE INHIBITORS. PART 3: THIOMORPHOLINETITL 2 SULFONAMIDE HYDROXAMATES.REF BIOORG.MED.CHEM.LETT. V. 16 1605 2006REFN ISSN 0960-894XPMID 16426848DOI 10.1016/J.BMCL.2005.12.020

Variant Set Distributions

ExAC Variants

Number Of Residues 259
Number Of SNVs 44
Number Of Permutations 21699
Optimal Distance Threshold 18.0
K Statistic 0.223
p-value 0.039

Mapped Variants

[+] ExAC Missense Variants